論文 - 横島 聡
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Intramolecular cycloaddition of nitrones in total synthesis of natural products. 査読有り
Yokoshima S
Natural product reports 2025年3月
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Total Synthesis of Melonine. 査読有り
Matsuyuki Y, Umekubo N, Yokoshima S
Organic letters 27 巻 ( 9 ) 頁: 2065 - 2068 2025年3月
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Total Synthesis of Putative Melognine 査読有り
Irie, Y; Yokoshima, S
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 146 巻 ( 14 ) 頁: 9526 - 9531 2024年3月
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Deep learning driven de novo drug design based on gastric proton pump structures. 査読有り
Abe K, Ozako M, Inukai M, Matsuyuki Y, Kitayama S, Kanai C, Nagai C, Gopalasingam CC, Gerle C, Shigematsu H, Umekubo N, Yokoshima S, Yoshimori A
Communications biology 6 巻 ( 1 ) 頁: 956 2023年9月
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Total syntheses of macleanine and lycoposerramine-S. 査読有り
Okuyama M, Umekubo N, Akimoto K, Shimizu T, Kubokoya K, Nakajima N, Nishiyama Y, Yokoshima S
Organic & biomolecular chemistry 21 巻 ( 31 ) 頁: 6289 - 6292 2023年8月
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Total Syntheses of Malettinins C and E. 査読有り
Umekubo N, Yokoshima S
Organic letters 25 巻 ( 24 ) 頁: 4530 - 4533 2023年6月
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Construction of the tetracyclic ring system of diterpene alkaloids via cationic [5 + 2] cycloaddition. 査読有り
Mizuno K, Nishiyama Y, Yokoshima S
Organic & biomolecular chemistry 21 巻 ( 22 ) 頁: 4587 - 4590 2023年6月
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Total Synthesis of Kopsone. 査読有り
Tomoya K, Komiya K, Nakajima D, Umekubo N, Yokoshima S
Organic letters 25 巻 ( 15 ) 頁: 2718 - 2721 2023年4月
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Fluorinated 2,6-Xylenesulfonyl Group: A Protective Group for Amines. 査読有り
Katayama Y, Watanabe K, Nishiyama Y, Yokoshima S
Organic letters 25 巻 ( 8 ) 頁: 1326 - 1330 2023年3月
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Convergent synthesis of the [5-7-6-3] tetracyclic core of premyrsinane diterpenes. 査読有り
Yoshinaga K, Yokoshima S
Organic & biomolecular chemistry 21 巻 ( 4 ) 頁: 724 - 727 2023年1月
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Construction of the [7-5-5] Tricyclic Core of Daphniphyllum Alkaloids via a Cationic Cascade Reaction. 査読有り
Nakajima D, Yokoshima S
Organic letters 24 巻 ( 51 ) 頁: 9520 - 9524 2022年12月
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Formal Synthesis of Ecteinascidin 743 via an Intramolecular Cascade Heck Reaction to Construct the Diazabicyclo[3.3.1]nonane Framework. 査読有り
Nakajima N, Yoshida E, Toma T, Nishiyama Y, Inoue M, Fukuyama T, Yokoshima S
Organic letters 24 巻 ( 44 ) 頁: 8228 - 8232 2022年11月
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Anticancer Approach Inspired by the Hepatotoxic Mechanism of Pyrrolizidine Alkaloids with Glycosylated Artificial Metalloenzymes. 査読有り
Kurimoto M, Chang TC, Nishiyama Y, Suzuki T, Dohmae N, Tanaka K, Yokoshima S
Angewandte Chemie (International ed. in English) 61 巻 ( 43 ) 頁: e202205541 2022年10月
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Photoinduced rearrangement of α-(2-nitrophenyl)ketones. 査読有り
Kitayama S, Shimizu H, Yokoshima S
Organic & biomolecular chemistry 20 巻 ( 40 ) 頁: 7896 - 7899 2022年10月
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Substitution of α-Azido Sulfones with Thiolates to Form α-Azido Sulfides. 査読有り
Katayama A, Jin Y, Nishiyama Y, Hosoya T, Yokoshima S
Organic letters 24 巻 ( 40 ) 頁: 7361 - 7365 2022年10月
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Synthetic Approach toward (-)-Tetrodotoxin via Construction of the Bicyclo[2.2.2]octane Skeleton 査読有り
Kobayashi Kazuki, Senoo Yoshiki, Toma Tatsuya, Fukuyama Tohru, Yokoshima Satoshi
SYNLETT 33 巻 ( 04 ) 頁: 391 - 395 2022年3月
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Photo-oxygenation by a biocompatible catalyst reduces amyloid-β levels in Alzheimer's disease mice. 査読有り
Ozawa S, Hori Y, Shimizu Y, Taniguchi A, Suzuki T, Wang W, Chiu YW, Koike R, Yokoshima S, Fukuyama T, Takatori S, Sohma Y, Kanai M, Tomita T
Brain : a journal of neurology 144 巻 ( 6 ) 頁: 1884 - 1897 2021年7月
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Total Synthesis of Haliclonin A. 査読有り
Jin Y, Orihara K, Kawagishi F, Toma T, Fukuyama T, Yokoshima S
Angewandte Chemie (International ed. in English) 60 巻 ( 17 ) 頁: 9666 - 9671 2021年4月
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Nitrone Formation by Reaction of an Enolate with a Nitro Group. 査読有り
Shimizu H, Yoshinaga K, Yokoshima S
Organic letters 23 巻 ( 7 ) 頁: 2704 - 2709 2021年4月
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A novel translation inhibitor, mersicarpine, inhibits S-phase progression and induces apoptosis in HL60 cells. 査読有り
Shiobara T, Nagumo Y, Nakajima R, Fukuyama T, Yokoshima S, Usui T
Bioscience, biotechnology, and biochemistry 85 巻 ( 1 ) 頁: 92 - 96 2021年1月
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Synthesis of 2-Azabicyclo[3.3.1]nonanes: Lessons from Synthetic Studies of Macrocyclic Diamine Alkaloids 招待有り 査読有り
Yokoshima Satoshi
CHEMISTRY LETTERS 50 巻 ( 1 ) 頁: 96 - 102 2021年1月
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Copper-Mediated Conversion of Alkynes into Nitriles via Iodotriazoles. 査読有り
Kori R, Murakami K, Nishiyama Y, Toma T, Yokoshima S
Chemical & pharmaceutical bulletin 69 巻 ( 3 ) 頁: 278 - 280 2021年
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SYNTHETIC STUDIES ON DENSANINS: STEREOSELECTIVE CONSTRUCTION OF A PYRROLIDINE RING CONTAINING A QUATERNARY CARBON 査読有り
Ueda Kyosuke, Yokoshima Satoshi
HETEROCYCLES 103 巻 ( 1 ) 頁: 172 - 176 2021年
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Synthesis of Polycyclic Natural Products through Skeletal Rearrangement 招待有り 査読有り
Yokoshima Satoshi
SYNLETT 31 巻 ( 20 ) 頁: 1967 - 1975 2020年12月
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Structure-Activity Relationship Study of Majusculamides A and B and Their Analogues on Osteogenic Activity. 査読有り
Natsume N, Ozaki K, Nakajima D, Yokoshima S, Teruya T
Journal of natural products 83 巻 ( 8 ) 頁: 2477 - 2482 2020年8月
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Semipinacol Rearrangement Induced by Cleavage of Dibromocyclopropane 査読有り
Kurimoto Michitaka, Nakajima Daisuke, Nishiyama Yoshitake, Yokoshima Satoshi
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY 2020 巻 ( 27 ) 頁: 4108 - 4111 2020年7月
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Total Synthesis of Tetrodotoxin. 査読有り
Murakami K, Toma T, Fukuyama T, Yokoshima S
Angewandte Chemie (International ed. in English) 59 巻 ( 15 ) 頁: 6253 - 6257 2020年4月
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Synthetic Studies on Bilobalide
Shiogai Akihiro, Toma Tatsuya, Yokoshima Satoshi
SYNLETT 31 巻 ( 3 ) 頁: 290 - 294 2020年2月
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An artificial metalloenzyme biosensor can detect ethylene gas in fruits and Arabidopsis leaves.
Vong K, Eda S, Kadota Y, Nasibullin I, Wakatake T, Yokoshima S, Shirasu K, Tanaka K
Nature communications 10 巻 ( 1 ) 頁: 5746 2019年12月
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Synthesis of Majusculamides A and B 査読有り
Nakajima Daisuke, Sueyoshi Kosuke, Orihara Kensuke, Teruya Toshiaki, Yokoshima Satoshi
SYNLETT 30 巻 ( 8 ) 頁: 924 - 927 2019年5月
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PREFACE TO HETEROCYCLES ISSUE HONORING THE 70TH BIRTHDAY OF PROFESSOR TOHRU FUKUYAMA
Yokoshima Satoshi
HETEROCYCLES 99 巻 ( 1 ) 頁: 1 - 3 2019年4月
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Synthetic Studies of Isoschizogamine: Alternative Preparation of the Key Intermediate.
Hayashi N, Miura Y, Yokoshima S, Fukuyama T
Chemical & pharmaceutical bulletin 67 巻 ( 1 ) 頁: 64 - 70 2019年1月
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天然物合成がもたらす新たな骨格構築と創薬 招待有り 査読有り
横島 聡
MEDCHEM NEWS 29 巻 ( 4 ) 頁: 178 - 182 2019年
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Total Synthesis of Lycoposerramine-R
Watanabe Shinya, Ishikawa Masatsugu, Nomura Toshimune, Fukuyama Tohru, Yokoshima Satoshi
SYNLETT 29 巻 ( 18 ) 頁: 2377-2380 2018年11月
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Synthetic Studies of the Daphniphyllum Alkaloids: A Cooperative Reaction of Proximal Functional Groups Forming a Tetracyclic System.
Yamada R, Fukuyama T, Yokoshima S
Organic letters 20 巻 ( 15 ) 頁: 4504 - 4506 2018年8月
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A small-molecule inhibitor of SOD1-Derlin-1 interaction ameliorates pathology in an ALS mouse model.
Tsuburaya N, Homma K, Higuchi T, Balia A, Yamakoshi H, Shibata N, Nakamura S, Nakagawa H, Ikeda SI, Umezawa N, Kato N, Yokoshima S, Shibuya M, Shimonishi M, Kojima H, Okabe T, Nagano T, Naguro I, Imamura K, Inoue H, Fujisawa T, Ichijo H
Nature communications 9 巻 ( 1 ) 頁: 2668 2018年7月
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Synthesis of the [7-5-5] tricyclic core of Daphniphyllum alkaloids.
Kitabayashi Y, Fukuyama T, Yokoshima S
Organic & biomolecular chemistry 16 巻 ( 19 ) 頁: 3556 - 3559 2018年5月
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Synthetic Studies of Haliclonin A: Construction of the 3-Azabicyclo[3.3.1]nonane Skeleton with a Bridge that Forms the 17-Membered Ring
Orihara Kensuke, Kawagishi Fumiki, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT 29 巻 ( 6 ) 頁: 769-772 2018年4月
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Total synthesis of (+)-lysergic acid 査読有り
Kanno Rentaro, Yokoshima Satoshi, Kanai Motomu, Fukuyama Tohru
JOURNAL OF ANTIBIOTICS 71 巻 ( 2 ) 頁: 240-247 2018年2月
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Total Synthesis of Huperzine R 査読有り
Nomura Toshimune, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 20 巻 ( 1 ) 頁: 119-121 2018年1月
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Synthesis of Cardiopetaline via a Wagner-Meerwein Rearrangement without Preactivation of the Pivotal Hydroxy Group 査読有り
Nishiyama Yoshitake, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 19 巻 ( 21 ) 頁: 5833-5835 2017年11月
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Synthesis of Lycopodium Alkaloids 査読有り
Yokoshima Satoshi
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN 75 巻 ( 10 ) 頁: 1035-1044 2017年10月
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Discovery of novel 2-(3-phenylpiperazin-1-yl)-pyrimidin-4-ones as glycogen synthase kinase-3 beta inhibitors 査読有り
Usui Yoshihiro, Uehara Fumiaki, Hiki Shinsuke, Watanabe Kazutoshi, Tanaka Hiroshi, Shouda Aya, Yokoshima Satoshi, Aritomo Keiichi, Adachi Takashi, Fukunaga Kenji, Sunada Shinji, Nabeno Mika, Saito Ken-Ichi, Eguchi Jun-ichi, Yamagami Keiji, Asano Shouichi, Tanaka Shinji, Yuki Satoshi, Yoshii Narihiko, Fujimura Masatake, Horikawa Takashi
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 27 巻 ( 16 ) 頁: 3726-3732 2017年8月
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Total Synthesis of Huperzine Q 査読有り
Tanimura Shun, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 19 巻 ( 13 ) 頁: 3684-3686 2017年7月
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High-throughput Screening of Small Molecule Inhibitors of the Streptococcus Quorum-sensing Signal Pathway 査読有り
Ishii Seiji, Fukui Kenji, Yokoshima Satoshi, Kumagai Kazuo, Beniyama Youko, Kodama Tetsuya, Fukuyama Tohru, Okabe Takayoshi, Nagano Tetsuo, Kojima Hirotatsu, Yano Takato
SCIENTIFIC REPORTS 7 巻 2017年6月
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Total Syntheses of Aurachins A and B 査読有り
Hattori Haruhiko, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 56 巻 ( 24 ) 頁: 6980-6983 2017年6月
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Total Synthesis of (-)-Morphine 査読有り
Umihara Hirotatsu, Yokoshima Satoshi, Inoue Masayuki, Fukuyama Tohru
CHEMISTRY-A EUROPEAN JOURNAL 23 巻 ( 29 ) 頁: 6993-6995 2017年5月
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Total Synthesis of (-)-Tetrodotoxin and 11-norTTX-6(R)-ol 査読有り
Maehara Tomoaki, Motoyama Keisuke, Toma Tatsuya, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 56 巻 ( 6 ) 頁: 1549-1552 2017年2月
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Total Synthesis of Lycopalhine A 査読有り
Ochi Yuji, Yokoshima Satoshi, Fukuyama Tohru
SYNTHESIS-STUTTGART 49 巻 ( 1 ) 頁: 96-114 2017年1月
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Chemical Transformation of an Intermediate in the Synthesis of Huperzine A, Leading to a Diverse Array of Molecules 査読有り
Yokoshima Satoshi, Ishikawa Masatsugu, Beniyama Youko, Fukuyama Tohru
CHEMICAL & PHARMACEUTICAL BULLETIN 64 巻 ( 10 ) 頁: 1528-1531 2016年10月
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Eudistomin C, an Antitumor and Antiviral Natural Product, Targets 40S Ribosome and Inhibits Protein Translation 査読有り
Ota Yu, Chinen Takumi, Yoshida Keisuke, Kudo Shun, Nagumo Yoko, Shiwa Yuh, Yamada Ryosuke, Umihara Hirotatsu, Iwasaki Kotaro, Masumoto Hiroshi, Yokoshima Satoshi, Yoshikawa Hirofumi, Fukuyama Tohru, Kobayashi Junichi, Usui Takeo
CHEMBIOCHEM 17 巻 ( 17 ) 頁: 1616-1620 2016年9月
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Morphological Evaluation of Nonlabeled Cells to Detect Stimulation of Nerve Growth Factor Expression by Lyconadin B 査読有り
Kawai Shun, Sasaki Hiroto, Okada Norihiro, Kanie Kei, Yokoshima Satoshi, Fukuyama Tohru, Honda Hiroyuki, Kato Ryuji
JOURNAL OF BIOMOLECULAR SCREENING 21 巻 ( 8 ) 頁: 795-803 2016年9月
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BIN1 regulates BACE1 intracellular trafficking and amyloid-beta production 査読有り
Miyagawa Toji, Ebinuma Ihori, Morohashi Yuichi, Hori Yukiko, Chang Mee Young, Hattori Haruhiko, Maehara Tomoaki, Yokoshima Satoshi, Fukuyama Tohru, Tsuji Shoji, Iwatsubo Takeshi, Prendergast George C., Tomita Taisuke
HUMAN MOLECULAR GENETICS 25 巻 ( 14 ) 頁: 2948-2958 2016年7月
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Conversion of Vindoline into 11-Mesyloxytabersonine 査読有り
Han-ya Yuki, Inui Tomohiko, Yokoshima Satoshi, Tokuyama Hidetoshi, Fukuyama Tohru
CHEMICAL & PHARMACEUTICAL BULLETIN 64 巻 ( 7 ) 頁: 800-804 2016年7月
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Total Synthesis of (-)-Cardiopetaline 査読有り
Nishiyama Yoshitake, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 18 巻 ( 10 ) 頁: 2359-2362 2016年5月
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Total Synthesis of (-)-Daphenylline 査読有り
Yamada Ryosuke, Adachi Yohei, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 55 巻 ( 20 ) 頁: 6067-6070 2016年5月
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Total Synthesis of Lycopalhine A 査読有り
Ochi Yuji, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 18 巻 ( 6 ) 頁: 1494-1496 2016年3月
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Synthetic Studies on Huperzine R: Construction of the 1-Azabicyclo[5.4.3]tetradec-6-ene Core 査読有り
Kumazaki Hiroshi, Nakajima Rie, Bessho Yuka, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT 26 巻 ( 15 ) 頁: 2131-2134 2015年9月
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Conversion of Ester Moieties to 4-Bromophenyl Groups via Electrocyclic Reaction of Dibromocyclopropanes 査読有り
Ueda Kyosuke, Umihara Hirotatsu, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 17 巻 ( 13 ) 頁: 3191-3193 2015年7月
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Synthetic Studies on Plakinidines 査読有り
Komori Takashi, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT 26 巻 ( 11 ) 頁: 1537-1540 2015年7月
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Formal Synthesis of Sarain A: Intramolecular Cycloaddition of an Eight-Membered Cyclic Nitrone to Construct the 2-Azabicyclo-[3.3.1]nonane Framework 査読有り
Higo Takuya, Ukegawa Tomoya, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 54 巻 ( 25 ) 頁: 7367-7370 2015年6月
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Asymmetric synthesis of 2-arylpiperazines 査読有り
Yokoshima Satoshi, Watanabe Kazutoshi, Uehara Fumiaki, Usui Yoshihiro, Tanaka Hiroshi
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 24 巻 ( 24 ) 頁: 5749-5751 2014年12月
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Synthesis of (-)-Oxycodone 査読有り
Kimishima Atsushi, Umihara Hirotatsu, Mizoguchi Akihiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 23 ) 頁: 6244-6247 2014年12月
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Total Synthesis of Lysergic Acid (vol 16, pg 1269, 2014) 査読有り
Umezaki Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 17 ) 頁: 4692-4692 2014年9月
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A Unified Strategy for Kainoid Synthesis 査読有り
Fujii Masaya, Yokoshima Satoshi, Fukuyama Tohru
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY ( 22 ) 頁: 4823-4836 2014年8月
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Allosteric regulation of gamma-secretase activity by a phenylimidazole-type gamma-secretase modulator 査読有り
Takeo Koji, Tanimura Shun, Shinoda Takehiro, Osawa Satoko, Zahariev Ivan Krasmirov, Takegami Naoki, Ishizuka-Katsura Yoshiko, Shinya Naoko, Takagi-Niidome Shizuka, Tominaga Aya, Ohsawa Noboru, Kimura-Someya Tomomi, Shirouzu Mikako, Yokoshima Satoshi, Yokoyama Shigeyuki, Fukuyama Tohru, Tomita Taisuke, Iwatsubo Takeshi
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA 111 巻 ( 29 ) 頁: 10544-10549 2014年7月
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New photocleavable linker: alpha-Thioacetophenone-type linker 査読有り
Yonezawa Hirotaka, Nishiyama Yoshitake, Takeo Koji, Iwatsubo Takeshi, Tomita Taisuke, Yokoshima Satoshi, Fukuyama Tohru
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 24 巻 ( 13 ) 頁: 2831-2833 2014年7月
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Total Synthesis of (-)-Lepistine 査読有り
Kitabayashi Yusuke, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 11 ) 頁: 2862-2864 2014年6月
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Total Synthesis of (-)-Lepenine 査読有り
Nishiyama Yoshitake, Han-ya Yuki, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 136 巻 ( 18 ) 頁: 6598-6601 2014年5月
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Total Synthesis of (-)-Mersicarpine (vol 132, pg 1236, 2010) 査読有り
Nakajima Rie, Ogino Tsuyoshi, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 136 巻 ( 15 ) 頁: 5816-5816 2014年4月
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Concise Total Synthesis of (+)-Lyconadin A (vol 133, pg 418, 2011) 査読有り
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 136 巻 ( 15 ) 頁: 5818-5818 2014年4月
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Total Synthesis of Ecteinascidin 743 (vol 135, pg 13684, 2013) 査読有り
Kawagishi Fumiki, Toma Tatsuya, Inui Tomohiko, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 136 巻 ( 15 ) 頁: 5815-5815 2014年4月
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Total Syntheses of Lyconadins A-C (vol 135, pg 3243, 2013) 査読有り
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 136 巻 ( 15 ) 頁: 5817-5817 2014年4月
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Correction of Synthetic Studies on Chartelline C: Stereoselective Construction of the Core Skeleton 査読有り
Iwasaki Kotaro, Kanno Rentaro, Morimoto Toshiharu, Yamashita Tohru, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 53 巻 ( 15 ) 頁: 3768-3768 2014年4月
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Total Synthesis of (-)-Huperzine A (vol 11, pg 5354, 2009) 査読有り
Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 4 ) 頁: 1270-1270 2014年2月
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(1-Nosyl-5-nitroindol-3-yl)methyl Ester: A Novel Protective Group for Carboxylic Acids (vol 10, pg 2601, 2008) 査読有り
Nishimura Takuya, Yamada Kouhei, Takebe Tohru, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 4 ) 頁: 1268-1268 2014年2月
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2-Pyridone Synthesis Using 2-(Phenylsulfinyl)acetamide (vol 15, pg 232, 2013) 査読有り
Fujii Masaya, Nishimura Takuya, Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 4 ) 頁: 1272-1272 2014年2月
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Total Synthesis of (-)-Histrionicotoxin (vol 13, pg 4466, 2011) 査読有り
Adachi Yohei, Kamei Noriyuki, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 4 ) 頁: 1273-1273 2014年2月
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Total Synthesis of Lysergic Acid (vol 15, pg 4230, 2013) 査読有り
Umezaki Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 16 巻 ( 4 ) 頁: 1269-1269 2014年2月
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Binding of longer A beta to transmembrane domain 1 of presenilin 1 impacts on A beta 42 generation 査読有り
Ohki Yu, Shimada Naoaki, Tominaga Aya, Osawa Satoko, Higo Takuya, Yokoshima Satoshi, Fukuyama Tohru, Tomita Taisuke, Iwatsubo Takeshi
MOLECULAR NEURODEGENERATION 9 巻 2014年1月
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Total Synthesis of Ecteinascidin 743 査読有り
Kawagishi Fumiki, Toma Tatsuya, Inui Tomohiko, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 135 巻 ( 37 ) 頁: 13684-13687 2013年9月
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Total Synthesis of Lysergic Acid 査読有り
Umezaki Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 15 巻 ( 16 ) 頁: 4230-4233 2013年8月
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Synthesis of Natural Products with Polycyclic Systems 査読有り
Yokoshima Satoshi
CHEMICAL & PHARMACEUTICAL BULLETIN 61 巻 ( 3 ) 頁: 251-257 2013年3月
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Effect of Helical Conformation and Side Chain Structure on gamma-Secretase Inhibition by beta-Peptide Foldamers: Insight into Substrate Recognition 査読有り
Imamura Yuki, Umezawa Naoki, Osawa Satoko, Shimada Naoaki, Higo Takuya, Yokoshima Satoshi, Fukuyama Tohru, Iwatsubo Takeshi, Kato Nobuki, Tomita Taisuke, Higuchi Tsunehiko
JOURNAL OF MEDICINAL CHEMISTRY 56 巻 ( 4 ) 頁: 1443-1454 2013年2月
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Total Syntheses of Lyconadins A-C 査読有り
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 135 巻 ( 8 ) 頁: 3243-3247 2013年2月
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2-Pyridone Synthesis Using 2-(Phenylsulfinyl)acetamide 査読有り
Fujii Masaya, Nishimura Takuya, Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 15 巻 ( 1 ) 頁: 232-234 2013年1月
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Activity-Dependent Proteolytic Cleavage of Neuroligin-1 査読有り
Suzuki Kunimichi, Hayashi Yukari, Nakahara Soichiro, Kumazaki Hiroshi, Prox Johannes, Horiuchi Keisuke, Zeng Mingshuo, Tanimura Shun, Nishiyama Yoshitake, Osawa Satoko, Sehara-Fujisawa Atsuko, Saftig Paul, Yokoshima Satoshi, Fukuyama Tohru, Matsuki Norio, Koyama Ryuta, Tomita Taisuke, Iwatsubo Takeshi
NEURON 76 巻 ( 2 ) 頁: 410-422 2012年10月
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Synthetic Studies toward Ecteinascidin 743 (Trabectedin) 査読有り
Imai Takahiro, Nakata Hiyoku, Yokoshima Satoshi, Fukuyama Tohru
SYNTHESIS-STUTTGART 44 巻 ( 17 ) 頁: 2743-2753 2012年9月
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Total Synthesis of (-)-Lemonomycin 査読有り
Yoshida Atsushi, Akaiwa Michinori, Asakawa Tomohiro, Hamashima Yoshitaka, Yokoshima Satoshi, Fukuyama Tohru, Kan Toshiyuki
CHEMISTRY-A EUROPEAN JOURNAL 18 巻 ( 36 ) 頁: 11192-11195 2012年9月
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Total Synthesis of (-)-Isoschizogamine 査読有り
Miura Yusuke, Hayashi Noriyuki, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 134 巻 ( 29 ) 頁: 11995-11997 2012年7月
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A Practical Preparation of Highly Versatile N-Acylpyrroles from 2,4,4-Trimethoxybutan-1-amine 査読有り
Maehara Tomoaki, Kanno Rentaro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 14 巻 ( 7 ) 頁: 1946-1948 2012年4月
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Total Synthesis of (-)-Anisatin 査読有り
Ogura Akihiro, Yamada Kohei, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 14 巻 ( 6 ) 頁: 1632-1635 2012年3月
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Identification of novel deoxyribofuranosyl indole antimicrobial agents 査読有り
Paudel Atmika, Hamamoto Hiroshi, Kobayashi Yoshihisa, Yokoshima Satoshi, Fukuyama Tohru, Sekimizu Kazuhisa
JOURNAL OF ANTIBIOTICS 65 巻 ( 2 ) 頁: 53-57 2012年2月
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Total synthesis of gelsemoxonine 査読有り
Shimokawa Jun, Harada Takaaki, Yokoshima Satoshi, Fukuyama Tohru
PURE AND APPLIED CHEMISTRY 84 巻 ( 7 ) 頁: 1643-1650 2012年
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Total Synthesis of (-)-Lycoposerramine-S 査読有り
Shimada Naoaki, Abe Yuzo, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 51 巻 ( 47 ) 頁: 11824-11826 2012年
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Synthetic Studies on Chartelline C: Stereoselective Construction of the Core Skeleton 査読有り
Iwasaki Kotaro, Kanno Rentaro, Morimoto Toshiharu, Yamashita Tohru, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 51 巻 ( 36 ) 頁: 9160-9163 2012年
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A Practical Synthesis of (-)-Kainic Acid 査読有り
Takita Satoshi, Yokoshima Satoshi, Fukuyama Tohru
SYNTHESIS-STUTTGART ( 23 ) 頁: 3848-3858 2011年12月
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Phenylpiperidine-type gamma-secretase modulators target the transmembrane domain 1 of presenilin 1 査読有り
Ohki Yu, Higo Takuya, Uemura Kengo, Shimada Naoaki, Osawa Satoko, Berezovska Oksana, Yokoshima Satoshi, Fukuyama Tohru, Tomita Taisuke, Iwatsubo Takeshi
EMBO JOURNAL 30 巻 ( 23 ) 頁: 4815-4824 2011年11月
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Total Synthesis of Gelsemoxonine 査読有り
Shimokawa Jun, Harada Takaaki, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 133 巻 ( 44 ) 頁: 17634-17637 2011年11月
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Practical synthesis of (-)-kainic acid 査読有り
Takita Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 242 巻 頁: . 2011年8月
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Total Synthesis of (-)-Histrionicotoxin 査読有り
Adachi Yohei, Kamei Noriyuki, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 13 巻 ( 16 ) 頁: 4446-4449 2011年8月
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Copper-Mediated Aryl Amination: In Situ Generation of an Active Copper(I) Species 査読有り
Komori Takashi, Satoh Nobuhiro, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT ( 13 ) 頁: 1859-1862 2011年8月
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Total Synthesis of (-)-Salinosporamide A 査読有り
Satoh Nobuhiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 13 巻 ( 12 ) 頁: 3028-3031 2011年6月
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BACE1 Activity Is Modulated by Cell-Associated Sphingosine-1-Phosphate 査読有り
Takasugi Nobumasa, Sasaki Tomoki, Suzuki Kunimichi, Osawa Satoko, Isshiki Hayato, Hori Yukiko, Shimada Naoaki, Higo Takuya, Yokoshima Satoshi, Fukuyama Tohru, Lee Virginia M. -Y., Trojanowski John Q., Tomita Taisuke, Iwatsubo Takeshi
JOURNAL OF NEUROSCIENCE 31 巻 ( 18 ) 頁: 6850-6857 2011年5月
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A Practical Synthesis of (-)-Kainic Acid 査読有り
Takita Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 13 巻 ( 8 ) 頁: 2068-2070 2011年4月
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Concise Total Synthesis of (+)-Lyconadin A 査読有り
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 133 巻 ( 3 ) 頁: 418-419 2011年1月
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Let's Challenge 査読有り
Yokoshima Satoshi
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN 68 巻 ( 12 ) 頁: 1323-1324 2010年12月
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Development of photoaffinity probes for gamma-secretase equipped with a nitrobenzenesulfonamide-type cleavable linker (vol 19, pg 6869, 2009) 査読有り
Yokoshima Satoshi, Abe Yuzo, Watanabe Naoto, Kita Yoichi, Kan Toshiyuki, Iwatsubo Takeshi, Tomita Taisuke, Fukuyama Tohru
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 20 巻 ( 5 ) 頁: 1798-1799 2010年3月
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Total Synthesis of (-)-Mersicarpine 査読有り
Nakajima Rie, Ogino Tsuyoshi, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 132 巻 ( 4 ) 頁: 1236-+ 2010年2月
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Total Synthesis of (-)-Morphine 査読有り
Koizumi Hifumi, Yokoshima Satoshi, Fukuyama Tohru
CHEMISTRY-AN ASIAN JOURNAL 5 巻 ( 10 ) 頁: 2192-2198 2010年
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Total Synthesis of (+)-Vinblastine: Control of the Stereochemistry at C18 ' 査読有り
Yokoshima Satoshi, Tokuyama Hidetoshi, Fukuyama Tohru
CHEMICAL RECORD 10 巻 ( 2 ) 頁: 101-118 2010年
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Development of photoaffinity probes for gamma-secretase equipped with a nitrobenzenesulfonamide-type cleavable linker 査読有り
Yokoshima Satoshi, Abe Yuzo, Watanabe Naoto, Kita Yoichi, Kan Toshiyuki, Iwatsubo Takeshi, Tomita Taisuke, Fukuyama Tohru
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 19 巻 ( 24 ) 頁: 6869-6871 2009年12月
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Total Synthesis of (-)-Huperzine A 査読有り
Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 11 巻 ( 22 ) 頁: 5354-5356 2009年11月
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A practical synthesis of (-)-oseltamivir 査読有り
Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
TETRAHEDRON 65 巻 ( 16 ) 頁: 3239-3245 2009年4月
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SYNTHETIC STUDIES TOWARD (+)-LYSERGIC ACID: CONSTRUCTION OF THE TETRACYCLIC ERGOLINE SKELETON 査読有り
Inoue Tohru, Yokoshima Satoshi, Fukuyama Tohru
HETEROCYCLES 79 巻 頁: 373-378 2009年4月
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TOTAL SYNTHESIS OF (+/-)-MORPHINE 査読有り
Uchida Kenji, Yokoshima Satoshi, Kan Toshiyuki, Fukuyama Tohru
HETEROCYCLES 77 巻 ( 2 ) 頁: 1219-1234 2009年2月
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A SIMPLE CHIRAL TEMPLATE FOR THE SYNTHESIS OF FUNCTIONALIZED alpha-ARYLGLYCINE DERIVATIVES 査読有り
Nakata Hiyoku, Imai Takahiro, Yokoshima Satoshi, Fukuyama Tohru
HETEROCYCLES 76 巻 ( 1 ) 頁: 747-757 2008年9月
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(1-nosyl-5-nitroindol-3-yl)methyl ester: A novel protective group for carboxylic acids 査読有り
Nishimura Takuya, Yamada Kouhei, Takebe Tohru, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS 10 巻 ( 12 ) 頁: 2601-2604 2008年6月
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Synthesis of eudistomin C and E: Improved preparation of the indole unit 査読有り
Yamagishi Hiroaki, Matsumoto Koji, Iwasaki Kotaro, Miyazaki Tohru, Yokoshima Satoshi, Tokuyama Hidetoshi, Fukuyama Tohru
ORGANIC LETTERS 10 巻 ( 12 ) 頁: 2369-2372 2008年6月
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Oseltamivir enhances hippocampal network synchronization 査読有り
Usami Atsushi, Sasaki Takuya, Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru, Yamatsugu Kenzo, Kanai Motomu, Shibasaki Masakatsu, Matsuki Norio, Ikegaya Yuji
JOURNAL OF PHARMACOLOGICAL SCIENCES 106 巻 ( 4 ) 頁: 659-662 2008年4月
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Oseltamivir induces spike synchronization in hippocampal networks 査読有り
Usami Atsushi, Sasaki Takuya, Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru, Yamatsugu Kenzo, Kanai Motomu, Shibasaki Masakatsu, Matsuki Norio, Ikegaya Yuji
JOURNAL OF PHARMACOLOGICAL SCIENCES 106 巻 頁: 173P-173P 2008年
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Synthesis of (+)-vinblastine and its analogues 査読有り
Miyazaki Tohru, Yokoshirna Satoshi, Simizu Siro, Osada Hiroyuki, Tokuyama Hidetoshi, Fukuyama Tohru
ORGANIC LETTERS 9 巻 ( 23 ) 頁: 4737-4740 2007年11月
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A practical synthesis of (-)-Oseltamivir 査読有り
Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 46 巻 ( 30 ) 頁: 5734-5736 2007年
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Diastereoselective synthesis of atropisomeric 3-(2-substituted aryl)quinazolin-4-ones and their stereochemical properties 査読有り
Tokitoh Takashi, Kobayashi Toshitake, Nakada Eisuke, Inoue Tohru, Yokoshima Satoshi, Takahashi Hideyo, Natsugari Hideaki
HETEROCYCLES 70 巻 頁: 93-+ 2006年12月
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Total synthesis of (+/-)-morphine 査読有り
Uchida Kenji, Yokoshima Satoshi, Kan Toshiyuki, Fukuyama Tohru
ORGANIC LETTERS 8 巻 ( 23 ) 頁: 5311-5313 2006年11月
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Synthesis of biotinylated photoaffinity probes based on arylsulfonamide gamma-secretase inhibitors 査読有り
Fuwa Haruhiko, Hiromoto Kenichi, Takahashi Yasuko, Yokoshima Satoshi, Kan Toshiyuki, Fukuyama Tohru, Iwatsubo Takeshi, Tomita Taisuke, Natsugari Hideaki
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 16 巻 ( 16 ) 頁: 4184-4189 2006年8月
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Novel gamma-secretase inhibitors discovered by library screening of in-house synthetic natural product intermediates 査読有り
Takahashi Y, Fuwa H, Kaneko A, Sasaki M, Yokoshima S, Koizumi H, Takebe T, Kan T, Iwatsubo T, Tomita T, Natsugari H, Fukuyama T
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 16 巻 ( 14 ) 頁: 3813-3816 2006年7月
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Stereocontrolled total synthesis of (+)-vincristine 査読有り
Kuboyama T, Yokoshima S, Tokuyama H, Fukuyama T
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA 101 巻 ( 33 ) 頁: 11966-11970 2004年8月
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A novel palladium-catalyzed coupling of thiol esters with 1-alkynes 査読有り
Tokuyama H, Miyazaki T, Yokoshima S, Fukuyama T
SYNLETT ( 10 ) 頁: 1512-1514 2003年8月
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Stereocontrolled total synthesis of (+)-vinblastine 査読有り
Yokoshima S, Ueda T, Kobayashi S, Sato A, Kuboyama T, Tokuyama H, Fukuyama T
PURE AND APPLIED CHEMISTRY 75 巻 ( 1 ) 頁: 29-38 2003年1月
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Reduction of ethanethiol esters to aldehydes 査読有り
Tokuyama H, Yokoshima S, Lin SC, Li LP, Fukuyama T
SYNTHESIS-STUTTGART ( 8 ) 頁: 1121-1123 2002年6月
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Stereocontrolled total synthesis of (+)-vinblastine 査読有り
Yokoshima S, Ueda T, Kobayashi S, Sato A, Kuboyama T, Tokuyama H, Fukuyama T
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 124 巻 ( 10 ) 頁: 2137-2139 2002年3月
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A novel oxidative transformation of alpha-aminonitriles to amides 査読有り
Yokoshima S, Kubo T, Tokuyama H, Fukuyama T
CHEMISTRY LETTERS ( 2 ) 頁: 122-123 2002年2月
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Dogger Bank Itch revisited: isolation of (2-hydroxyethyl) dimethylsulfoxonium chloride as a cytotoxic constituent from the marine sponge Theonella aff. mirabilis 査読有り
Warabi K, Nakao Y, Matsunaga S, Fukuyama T, Kan T, Yokoshima S, Fusetani N
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY B-BIOCHEMISTRY & MOLECULAR BIOLOGY 128 巻 ( 1 ) 頁: 27-30 2001年1月
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Enantioselective total synthesis of (+)-gelsemine: Determination of its absolute configuration 査読有り
Yokoshima S, Tokuyama H, Fukuyama T
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 39 巻 ( 22 ) 頁: 4073-4075 2000年
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A novel ketone synthesis by a palladium-catalyzed reaction of thiol esters and organozinc reagents 査読有り
Tokuyama H, Yokoshima S, Yamashita T, Fukuyama T
TETRAHEDRON LETTERS 39 巻 ( 20 ) 頁: 3189-3192 1998年5月
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Facile palladium-mediated conversion of ethanethiol esters to aldehydes and ketones 査読有り
Tokuyama H, Yokoshima S, Yamashita T, Lin SC, Li LP, Fukuyama T
JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY 9 巻 ( 4 ) 頁: 381-387 1998年