Papers - YOKOSHIMA Satoshi
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Furuhashi, K; Umekubo, N; Matsuyuki, Y; Yokoshima, S
ORGANIC LETTERS Vol. 27 ( 19 ) page: 4904 - 4908 2025.5
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Intramolecular cycloaddition of nitrones in total synthesis of natural products. Reviewed
Yokoshima S
Natural product reports 2025.3
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Total Synthesis of Melonine. Reviewed
Matsuyuki Y, Umekubo N, Yokoshima S
Organic letters Vol. 27 ( 9 ) page: 2065 - 2068 2025.3
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Total Synthesis of Putative Melognine. Reviewed
Vol. 146 ( 14 ) page: 9526 - 9531 2024.3
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Deep learning driven de novo drug design based on gastric proton pump structures. Reviewed
Abe K, Ozako M, Inukai M, Matsuyuki Y, Kitayama S, Kanai C, Nagai C, Gopalasingam CC, Gerle C, Shigematsu H, Umekubo N, Yokoshima S, Yoshimori A
Communications biology Vol. 6 ( 1 ) page: 956 2023.9
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Total syntheses of macleanine and lycoposerramine-S. Reviewed
Okuyama M, Umekubo N, Akimoto K, Shimizu T, Kubokoya K, Nakajima N, Nishiyama Y, Yokoshima S
Organic & biomolecular chemistry Vol. 21 ( 31 ) page: 6289 - 6292 2023.8
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Total Syntheses of Malettinins C and E. Reviewed
Umekubo N, Yokoshima S
Organic letters Vol. 25 ( 24 ) page: 4530 - 4533 2023.6
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Construction of the tetracyclic ring system of diterpene alkaloids via cationic [5 + 2] cycloaddition. Reviewed
Mizuno K, Nishiyama Y, Yokoshima S
Organic & biomolecular chemistry Vol. 21 ( 22 ) page: 4587 - 4590 2023.6
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Total Synthesis of Kopsone. Reviewed
Tomoya K, Komiya K, Nakajima D, Umekubo N, Yokoshima S
Organic letters Vol. 25 ( 15 ) page: 2718 - 2721 2023.4
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Fluorinated 2,6-Xylenesulfonyl Group: A Protective Group for Amines. Reviewed
Katayama Y, Watanabe K, Nishiyama Y, Yokoshima S
Organic letters Vol. 25 ( 8 ) page: 1326 - 1330 2023.3
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Convergent synthesis of the [5-7-6-3] tetracyclic core of premyrsinane diterpenes. Reviewed
Yoshinaga K, Yokoshima S
Organic & biomolecular chemistry Vol. 21 ( 4 ) page: 724 - 727 2023.1
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Construction of the [7-5-5] Tricyclic Core of Daphniphyllum Alkaloids via a Cationic Cascade Reaction. Reviewed
Nakajima D, Yokoshima S
Organic letters Vol. 24 ( 51 ) page: 9520 - 9524 2022.12
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Formal Synthesis of Ecteinascidin 743 via an Intramolecular Cascade Heck Reaction to Construct the Diazabicyclo[3.3.1]nonane Framework. Reviewed
Nakajima N, Yoshida E, Toma T, Nishiyama Y, Inoue M, Fukuyama T, Yokoshima S
Organic letters Vol. 24 ( 44 ) page: 8228 - 8232 2022.11
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Anticancer Approach Inspired by the Hepatotoxic Mechanism of Pyrrolizidine Alkaloids with Glycosylated Artificial Metalloenzymes. Reviewed
Kurimoto M, Chang TC, Nishiyama Y, Suzuki T, Dohmae N, Tanaka K, Yokoshima S
Angewandte Chemie (International ed. in English) Vol. 61 ( 43 ) page: e202205541 2022.10
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Photoinduced rearrangement of α-(2-nitrophenyl)ketones. Reviewed
Kitayama S, Shimizu H, Yokoshima S
Organic & biomolecular chemistry Vol. 20 ( 40 ) page: 7896 - 7899 2022.10
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Substitution of α-Azido Sulfones with Thiolates to Form α-Azido Sulfides. Reviewed
Katayama A, Jin Y, Nishiyama Y, Hosoya T, Yokoshima S
Organic letters Vol. 24 ( 40 ) page: 7361 - 7365 2022.10
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Synthetic Approach toward (-)-Tetrodotoxin via Construction of the Bicyclo[2.2.2]octane Skeleton Reviewed
Kobayashi Kazuki, Senoo Yoshiki, Toma Tatsuya, Fukuyama Tohru, Yokoshima Satoshi
SYNLETT Vol. 33 ( 04 ) page: 391 - 395 2022.3
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Photo-oxygenation by a biocompatible catalyst reduces amyloid-β levels in Alzheimer's disease mice. Reviewed
Ozawa S, Hori Y, Shimizu Y, Taniguchi A, Suzuki T, Wang W, Chiu YW, Koike R, Yokoshima S, Fukuyama T, Takatori S, Sohma Y, Kanai M, Tomita T
Brain : a journal of neurology Vol. 144 ( 6 ) page: 1884 - 1897 2021.7
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Total Synthesis of Haliclonin A. Reviewed
Jin Y, Orihara K, Kawagishi F, Toma T, Fukuyama T, Yokoshima S
Angewandte Chemie (International ed. in English) Vol. 60 ( 17 ) page: 9666 - 9671 2021.4
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Nitrone Formation by Reaction of an Enolate with a Nitro Group. Reviewed
Shimizu H, Yoshinaga K, Yokoshima S
Organic letters Vol. 23 ( 7 ) page: 2704 - 2709 2021.4
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A novel translation inhibitor, mersicarpine, inhibits S-phase progression and induces apoptosis in HL60 cells. Reviewed
Shiobara T, Nagumo Y, Nakajima R, Fukuyama T, Yokoshima S, Usui T
Bioscience, biotechnology, and biochemistry Vol. 85 ( 1 ) page: 92 - 96 2021.1
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Synthesis of 2-Azabicyclo[3.3.1]nonanes: Lessons from Synthetic Studies of Macrocyclic Diamine Alkaloids Invited Reviewed
Yokoshima Satoshi
CHEMISTRY LETTERS Vol. 50 ( 1 ) page: 96 - 102 2021.1
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Copper-Mediated Conversion of Alkynes into Nitriles via Iodotriazoles. Reviewed
Kori R, Murakami K, Nishiyama Y, Toma T, Yokoshima S
Chemical & pharmaceutical bulletin Vol. 69 ( 3 ) page: 278 - 280 2021
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SYNTHETIC STUDIES ON DENSANINS: STEREOSELECTIVE CONSTRUCTION OF A PYRROLIDINE RING CONTAINING A QUATERNARY CARBON Reviewed
Ueda Kyosuke, Yokoshima Satoshi
HETEROCYCLES Vol. 103 ( 1 ) page: 172 - 176 2021
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Synthesis of Polycyclic Natural Products through Skeletal Rearrangement Invited Reviewed
Yokoshima Satoshi
SYNLETT Vol. 31 ( 20 ) page: 1967 - 1975 2020.12
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Structure-Activity Relationship Study of Majusculamides A and B and Their Analogues on Osteogenic Activity Reviewed
Natsume Noriyuki, Ozaki Kaori, Nakajima Daisuke, Yokoshima Satoshi, Teruya Toshiaki
JOURNAL OF NATURAL PRODUCTS Vol. 83 ( 8 ) page: 2477 - 2482 2020.8
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Semipinacol Rearrangement Induced by Cleavage of Dibromocyclopropane Reviewed
Kurimoto Michitaka, Nakajima Daisuke, Nishiyama Yoshitake, Yokoshima Satoshi
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY Vol. 2020 ( 27 ) page: 4108 - 4111 2020.7
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Total Synthesis of Tetrodotoxin Reviewed
Murakami Keigo, Toma Tatsuya, Fukuyama Tohru, Yokoshima Satoshi
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 59 ( 15 ) page: 6253 - 6257 2020.4
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Synthetic Studies on Bilobalide
Shiogai Akihiro, Toma Tatsuya, Yokoshima Satoshi
SYNLETT Vol. 31 ( 3 ) page: 290 - 294 2020.2
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An artificial metalloenzyme biosensor can detect ethylene gas in fruits and Arabidopsis leaves
Vong Kenward, Eda Shohei, Kadota Yasuhiro, Nasibullin Igor, Wakatake Takanori, Yokoshima Satoshi, Shirasu Ken, Tanaka Katsunori
NATURE COMMUNICATIONS Vol. 10 ( 1 ) page: 5746 2019.12
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Synthesis of Majusculamides A and B Reviewed
Nakajima Daisuke, Sueyoshi Kosuke, Orihara Kensuke, Teruya Toshiaki, Yokoshima Satoshi
SYNLETT Vol. 30 ( 8 ) page: 924 - 927 2019.5
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PREFACE TO HETEROCYCLES ISSUE HONORING THE 70TH BIRTHDAY OF PROFESSOR TOHRU FUKUYAMA
Yokoshima Satoshi
HETEROCYCLES Vol. 99 ( 1 ) page: 1 - 3 2019.4
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Synthetic Studies of Isoschizogamine: Alternative Preparation of the Key Intermediate.
Hayashi N, Miura Y, Yokoshima S, Fukuyama T
Chemical & pharmaceutical bulletin Vol. 67 ( 1 ) page: 64 - 70 2019.1
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天然物合成がもたらす新たな骨格構築と創薬 Invited Reviewed
横島 聡
MEDCHEM NEWS Vol. 29 ( 4 ) page: 178 - 182 2019
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Total Synthesis of Lycoposerramine-R
Watanabe Shinya, Ishikawa Masatsugu, Nomura Toshimune, Fukuyama Tohru, Yokoshima Satoshi
SYNLETT Vol. 29 ( 18 ) page: 2377-2380 2018.11
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Synthetic Studies of the Daphniphyllum Alkaloids: A Cooperative Reaction of Proximal Functional Groups Forming a Tetracyclic System
Yamada Ryosuke, Fukuyama Tohru, Yokoshima Satoshi
ORGANIC LETTERS Vol. 20 ( 15 ) page: 4504 - 4506 2018.8
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A small-molecule inhibitor of SOD1-Derlin-1 interaction ameliorates pathology in an ALS mouse model
Tsuburaya Naomi, Homma Kengo, Higuchi Tsunehiko, Balia Andrii, Yamakoshi Hiroyuki, Shibata Norio, Nakamura Seiichi, Nakagawa Hidehiko, Ikeda Shin-ichi, Umezawa Naoki, Kato Nobuki, Yokoshima Satoshi, Shibuya Masatoshi, Shimonishi Manabu, Kojima Hirotatsu, Okabe Takayoshi, Nagano Tetsuo, Naguro Isao, Imamura Keiko, Inoue Haruhisa, Fujisawa Takao, Ichijo Hidenori
NATURE COMMUNICATIONS Vol. 9 ( 1 ) page: 2668 2018.7
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Synthesis of the [7-5-5] tricyclic core of Daphniphyllum alkaloids
Kitabayashi Yusuke, Fukuyama Tohru, Yokoshima Satoshi
ORGANIC & BIOMOLECULAR CHEMISTRY Vol. 16 ( 19 ) page: 3556 - 3559 2018.5
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Synthetic Studies of Haliclonin A: Construction of the 3-Azabicyclo[3.3.1]nonane Skeleton with a Bridge that Forms the 17-Membered Ring
Orihara Kensuke, Kawagishi Fumiki, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT Vol. 29 ( 6 ) page: 769-772 2018.4
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Total synthesis of (+)-lysergic acid Reviewed
Kanno Rentaro, Yokoshima Satoshi, Kanai Motomu, Fukuyama Tohru
JOURNAL OF ANTIBIOTICS Vol. 71 ( 2 ) page: 240-247 2018.2
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Total Synthesis of Huperzine R Reviewed
Nomura Toshimune, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 20 ( 1 ) page: 119-121 2018.1
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Synthesis of Cardiopetaline via a Wagner-Meerwein Rearrangement without Preactivation of the Pivotal Hydroxy Group Reviewed
Nishiyama Yoshitake, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 19 ( 21 ) page: 5833-5835 2017.11
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Synthesis of Lycopodium Alkaloids Reviewed
Yokoshima Satoshi
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN Vol. 75 ( 10 ) page: 1035-1044 2017.10
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Discovery of novel 2-(3-phenylpiperazin-1-yl)-pyrimidin-4-ones as glycogen synthase kinase-3 beta inhibitors Reviewed
Usui Yoshihiro, Uehara Fumiaki, Hiki Shinsuke, Watanabe Kazutoshi, Tanaka Hiroshi, Shouda Aya, Yokoshima Satoshi, Aritomo Keiichi, Adachi Takashi, Fukunaga Kenji, Sunada Shinji, Nabeno Mika, Saito Ken-Ichi, Eguchi Jun-ichi, Yamagami Keiji, Asano Shouichi, Tanaka Shinji, Yuki Satoshi, Yoshii Narihiko, Fujimura Masatake, Horikawa Takashi
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 27 ( 16 ) page: 3726-3732 2017.8
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Total Synthesis of Huperzine Q Reviewed
Tanimura Shun, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 19 ( 13 ) page: 3684-3686 2017.7
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High-throughput Screening of Small Molecule Inhibitors of the Streptococcus Quorum-sensing Signal Pathway Reviewed
Ishii Seiji, Fukui Kenji, Yokoshima Satoshi, Kumagai Kazuo, Beniyama Youko, Kodama Tetsuya, Fukuyama Tohru, Okabe Takayoshi, Nagano Tetsuo, Kojima Hirotatsu, Yano Takato
SCIENTIFIC REPORTS Vol. 7 2017.6
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Total Syntheses of Aurachins A and B Reviewed
Hattori Haruhiko, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 56 ( 24 ) page: 6980-6983 2017.6
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Total Synthesis of (-)-Morphine Reviewed
Umihara Hirotatsu, Yokoshima Satoshi, Inoue Masayuki, Fukuyama Tohru
CHEMISTRY-A EUROPEAN JOURNAL Vol. 23 ( 29 ) page: 6993-6995 2017.5
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Total Synthesis of (-)-Tetrodotoxin and 11-norTTX-6(R)-ol Reviewed
Maehara Tomoaki, Motoyama Keisuke, Toma Tatsuya, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 56 ( 6 ) page: 1549-1552 2017.2
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Total Synthesis of Lycopalhine A Reviewed
Ochi Yuji, Yokoshima Satoshi, Fukuyama Tohru
SYNTHESIS-STUTTGART Vol. 49 ( 1 ) page: 96-114 2017.1
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Chemical Transformation of an Intermediate in the Synthesis of Huperzine A, Leading to a Diverse Array of Molecules Reviewed
Yokoshima Satoshi, Ishikawa Masatsugu, Beniyama Youko, Fukuyama Tohru
CHEMICAL & PHARMACEUTICAL BULLETIN Vol. 64 ( 10 ) page: 1528-1531 2016.10
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Eudistomin C, an Antitumor and Antiviral Natural Product, Targets 40S Ribosome and Inhibits Protein Translation Reviewed
Ota Yu, Chinen Takumi, Yoshida Keisuke, Kudo Shun, Nagumo Yoko, Shiwa Yuh, Yamada Ryosuke, Umihara Hirotatsu, Iwasaki Kotaro, Masumoto Hiroshi, Yokoshima Satoshi, Yoshikawa Hirofumi, Fukuyama Tohru, Kobayashi Junichi, Usui Takeo
CHEMBIOCHEM Vol. 17 ( 17 ) page: 1616-1620 2016.9
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Morphological Evaluation of Nonlabeled Cells to Detect Stimulation of Nerve Growth Factor Expression by Lyconadin B Reviewed
Kawai Shun, Sasaki Hiroto, Okada Norihiro, Kanie Kei, Yokoshima Satoshi, Fukuyama Tohru, Honda Hiroyuki, Kato Ryuji
JOURNAL OF BIOMOLECULAR SCREENING Vol. 21 ( 8 ) page: 795-803 2016.9
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BIN1 regulates BACE1 intracellular trafficking and amyloid-beta production Reviewed
Miyagawa Toji, Ebinuma Ihori, Morohashi Yuichi, Hori Yukiko, Chang Mee Young, Hattori Haruhiko, Maehara Tomoaki, Yokoshima Satoshi, Fukuyama Tohru, Tsuji Shoji, Iwatsubo Takeshi, Prendergast George C., Tomita Taisuke
HUMAN MOLECULAR GENETICS Vol. 25 ( 14 ) page: 2948-2958 2016.7
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Conversion of Vindoline into 11-Mesyloxytabersonine Reviewed
Han-ya Yuki, Inui Tomohiko, Yokoshima Satoshi, Tokuyama Hidetoshi, Fukuyama Tohru
CHEMICAL & PHARMACEUTICAL BULLETIN Vol. 64 ( 7 ) page: 800-804 2016.7
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Total Synthesis of (-)-Cardiopetaline Reviewed
Nishiyama Yoshitake, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 18 ( 10 ) page: 2359-2362 2016.5
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Total Synthesis of (-)-Daphenylline Reviewed
Yamada Ryosuke, Adachi Yohei, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 55 ( 20 ) page: 6067-6070 2016.5
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Total Synthesis of Lycopalhine A Reviewed
Ochi Yuji, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 18 ( 6 ) page: 1494-1496 2016.3
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Synthetic Studies on Huperzine R: Construction of the 1-Azabicyclo[5.4.3]tetradec-6-ene Core Reviewed
Kumazaki Hiroshi, Nakajima Rie, Bessho Yuka, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT Vol. 26 ( 15 ) page: 2131-2134 2015.9
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Conversion of Ester Moieties to 4-Bromophenyl Groups via Electrocyclic Reaction of Dibromocyclopropanes Reviewed
Ueda Kyosuke, Umihara Hirotatsu, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 17 ( 13 ) page: 3191-3193 2015.7
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Synthetic Studies on Plakinidines Reviewed
Komori Takashi, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT Vol. 26 ( 11 ) page: 1537-1540 2015.7
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Formal Synthesis of Sarain A: Intramolecular Cycloaddition of an Eight-Membered Cyclic Nitrone to Construct the 2-Azabicyclo-[3.3.1]nonane Framework Reviewed
Higo Takuya, Ukegawa Tomoya, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 54 ( 25 ) page: 7367-7370 2015.6
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Asymmetric synthesis of 2-arylpiperazines Reviewed
Yokoshima Satoshi, Watanabe Kazutoshi, Uehara Fumiaki, Usui Yoshihiro, Tanaka Hiroshi
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 24 ( 24 ) page: 5749-5751 2014.12
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Synthesis of (-)-Oxycodone Reviewed
Kimishima Atsushi, Umihara Hirotatsu, Mizoguchi Akihiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 23 ) page: 6244-6247 2014.12
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Total Synthesis of Lysergic Acid (vol 16, pg 1269, 2014) Reviewed
Umezaki Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 17 ) page: 4692-4692 2014.9
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A Unified Strategy for Kainoid Synthesis Reviewed
Fujii Masaya, Yokoshima Satoshi, Fukuyama Tohru
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY ( 22 ) page: 4823-4836 2014.8
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Allosteric regulation of gamma-secretase activity by a phenylimidazole-type gamma-secretase modulator Reviewed
Takeo Koji, Tanimura Shun, Shinoda Takehiro, Osawa Satoko, Zahariev Ivan Krasmirov, Takegami Naoki, Ishizuka-Katsura Yoshiko, Shinya Naoko, Takagi-Niidome Shizuka, Tominaga Aya, Ohsawa Noboru, Kimura-Someya Tomomi, Shirouzu Mikako, Yokoshima Satoshi, Yokoyama Shigeyuki, Fukuyama Tohru, Tomita Taisuke, Iwatsubo Takeshi
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA Vol. 111 ( 29 ) page: 10544-10549 2014.7
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New photocleavable linker: alpha-Thioacetophenone-type linker Reviewed
Yonezawa Hirotaka, Nishiyama Yoshitake, Takeo Koji, Iwatsubo Takeshi, Tomita Taisuke, Yokoshima Satoshi, Fukuyama Tohru
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 24 ( 13 ) page: 2831-2833 2014.7
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Total Synthesis of (-)-Lepistine Reviewed
Kitabayashi Yusuke, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 11 ) page: 2862-2864 2014.6
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Total Synthesis of (-)-Lepenine Reviewed
Nishiyama Yoshitake, Han-ya Yuki, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 136 ( 18 ) page: 6598-6601 2014.5
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Total Synthesis of (-)-Mersicarpine (vol 132, pg 1236, 2010) Reviewed
Nakajima Rie, Ogino Tsuyoshi, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 136 ( 15 ) page: 5816-5816 2014.4
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Concise Total Synthesis of (+)-Lyconadin A (vol 133, pg 418, 2011) Reviewed
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 136 ( 15 ) page: 5818-5818 2014.4
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Total Synthesis of Ecteinascidin 743 (vol 135, pg 13684, 2013) Reviewed
Kawagishi Fumiki, Toma Tatsuya, Inui Tomohiko, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 136 ( 15 ) page: 5815-5815 2014.4
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Total Syntheses of Lyconadins A-C (vol 135, pg 3243, 2013) Reviewed
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 136 ( 15 ) page: 5817-5817 2014.4
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Correction of Synthetic Studies on Chartelline C: Stereoselective Construction of the Core Skeleton Reviewed
Iwasaki Kotaro, Kanno Rentaro, Morimoto Toshiharu, Yamashita Tohru, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 53 ( 15 ) page: 3768-3768 2014.4
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Total Synthesis of (-)-Huperzine A (vol 11, pg 5354, 2009) Reviewed
Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 4 ) page: 1270-1270 2014.2
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(1-Nosyl-5-nitroindol-3-yl)methyl Ester: A Novel Protective Group for Carboxylic Acids (vol 10, pg 2601, 2008) Reviewed
Nishimura Takuya, Yamada Kouhei, Takebe Tohru, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 4 ) page: 1268-1268 2014.2
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2-Pyridone Synthesis Using 2-(Phenylsulfinyl)acetamide (vol 15, pg 232, 2013) Reviewed
Fujii Masaya, Nishimura Takuya, Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 4 ) page: 1272-1272 2014.2
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Total Synthesis of (-)-Histrionicotoxin (vol 13, pg 4466, 2011) Reviewed
Adachi Yohei, Kamei Noriyuki, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 4 ) page: 1273-1273 2014.2
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Total Synthesis of Lysergic Acid (vol 15, pg 4230, 2013) Reviewed
Umezaki Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 16 ( 4 ) page: 1269-1269 2014.2
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Binding of longer A beta to transmembrane domain 1 of presenilin 1 impacts on A beta 42 generation Reviewed
Ohki Yu, Shimada Naoaki, Tominaga Aya, Osawa Satoko, Higo Takuya, Yokoshima Satoshi, Fukuyama Tohru, Tomita Taisuke, Iwatsubo Takeshi
MOLECULAR NEURODEGENERATION Vol. 9 2014.1
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Total Synthesis of Ecteinascidin 743 Reviewed
Kawagishi Fumiki, Toma Tatsuya, Inui Tomohiko, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 135 ( 37 ) page: 13684-13687 2013.9
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Total Synthesis of Lysergic Acid Reviewed
Umezaki Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 15 ( 16 ) page: 4230-4233 2013.8
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Synthesis of Natural Products with Polycyclic Systems Reviewed
Yokoshima Satoshi
CHEMICAL & PHARMACEUTICAL BULLETIN Vol. 61 ( 3 ) page: 251-257 2013.3
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Effect of Helical Conformation and Side Chain Structure on gamma-Secretase Inhibition by beta-Peptide Foldamers: Insight into Substrate Recognition Reviewed
Imamura Yuki, Umezawa Naoki, Osawa Satoko, Shimada Naoaki, Higo Takuya, Yokoshima Satoshi, Fukuyama Tohru, Iwatsubo Takeshi, Kato Nobuki, Tomita Taisuke, Higuchi Tsunehiko
JOURNAL OF MEDICINAL CHEMISTRY Vol. 56 ( 4 ) page: 1443-1454 2013.2
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Total Syntheses of Lyconadins A-C Reviewed
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 135 ( 8 ) page: 3243-3247 2013.2
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2-Pyridone Synthesis Using 2-(Phenylsulfinyl)acetamide Reviewed
Fujii Masaya, Nishimura Takuya, Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 15 ( 1 ) page: 232-234 2013.1
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Activity-Dependent Proteolytic Cleavage of Neuroligin-1 Reviewed
Suzuki Kunimichi, Hayashi Yukari, Nakahara Soichiro, Kumazaki Hiroshi, Prox Johannes, Horiuchi Keisuke, Zeng Mingshuo, Tanimura Shun, Nishiyama Yoshitake, Osawa Satoko, Sehara-Fujisawa Atsuko, Saftig Paul, Yokoshima Satoshi, Fukuyama Tohru, Matsuki Norio, Koyama Ryuta, Tomita Taisuke, Iwatsubo Takeshi
NEURON Vol. 76 ( 2 ) page: 410-422 2012.10
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Synthetic Studies toward Ecteinascidin 743 (Trabectedin) Reviewed
Imai Takahiro, Nakata Hiyoku, Yokoshima Satoshi, Fukuyama Tohru
SYNTHESIS-STUTTGART Vol. 44 ( 17 ) page: 2743-2753 2012.9
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Total Synthesis of (-)-Lemonomycin Reviewed
Yoshida Atsushi, Akaiwa Michinori, Asakawa Tomohiro, Hamashima Yoshitaka, Yokoshima Satoshi, Fukuyama Tohru, Kan Toshiyuki
CHEMISTRY-A EUROPEAN JOURNAL Vol. 18 ( 36 ) page: 11192-11195 2012.9
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Total Synthesis of (-)-Isoschizogamine Reviewed
Miura Yusuke, Hayashi Noriyuki, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 134 ( 29 ) page: 11995-11997 2012.7
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A Practical Preparation of Highly Versatile N-Acylpyrroles from 2,4,4-Trimethoxybutan-1-amine Reviewed
Maehara Tomoaki, Kanno Rentaro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 14 ( 7 ) page: 1946-1948 2012.4
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Total Synthesis of (-)-Anisatin Reviewed
Ogura Akihiro, Yamada Kohei, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 14 ( 6 ) page: 1632-1635 2012.3
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Identification of novel deoxyribofuranosyl indole antimicrobial agents Reviewed
Paudel Atmika, Hamamoto Hiroshi, Kobayashi Yoshihisa, Yokoshima Satoshi, Fukuyama Tohru, Sekimizu Kazuhisa
JOURNAL OF ANTIBIOTICS Vol. 65 ( 2 ) page: 53-57 2012.2
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Total synthesis of gelsemoxonine Reviewed
Shimokawa Jun, Harada Takaaki, Yokoshima Satoshi, Fukuyama Tohru
PURE AND APPLIED CHEMISTRY Vol. 84 ( 7 ) page: 1643-1650 2012
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Synthetic Studies on Chartelline C: Stereoselective Construction of the Core Skeleton Reviewed
Iwasaki Kotaro, Kanno Rentaro, Morimoto Toshiharu, Yamashita Tohru, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 51 ( 36 ) page: 9160-9163 2012
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Total Synthesis of (-)-Lycoposerramine-S Reviewed
Shimada Naoaki, Abe Yuzo, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 51 ( 47 ) page: 11824-11826 2012
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A Practical Synthesis of (-)-Kainic Acid Reviewed
Takita Satoshi, Yokoshima Satoshi, Fukuyama Tohru
SYNTHESIS-STUTTGART ( 23 ) page: 3848-3858 2011.12
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Phenylpiperidine-type gamma-secretase modulators target the transmembrane domain 1 of presenilin 1 Reviewed
Ohki Yu, Higo Takuya, Uemura Kengo, Shimada Naoaki, Osawa Satoko, Berezovska Oksana, Yokoshima Satoshi, Fukuyama Tohru, Tomita Taisuke, Iwatsubo Takeshi
EMBO JOURNAL Vol. 30 ( 23 ) page: 4815-4824 2011.11
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Total Synthesis of Gelsemoxonine Reviewed
Shimokawa Jun, Harada Takaaki, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 133 ( 44 ) page: 17634-17637 2011.11
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Practical synthesis of (-)-kainic acid Reviewed
Takita Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY Vol. 242 page: . 2011.8
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Total Synthesis of (-)-Histrionicotoxin Reviewed
Adachi Yohei, Kamei Noriyuki, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 13 ( 16 ) page: 4446-4449 2011.8
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Copper-Mediated Aryl Amination: In Situ Generation of an Active Copper(I) Species Reviewed
Komori Takashi, Satoh Nobuhiro, Yokoshima Satoshi, Fukuyama Tohru
SYNLETT ( 13 ) page: 1859-1862 2011.8
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Total Synthesis of (-)-Salinosporamide A Reviewed
Satoh Nobuhiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 13 ( 12 ) page: 3028-3031 2011.6
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BACE1 Activity Is Modulated by Cell-Associated Sphingosine-1-Phosphate Reviewed
Takasugi Nobumasa, Sasaki Tomoki, Suzuki Kunimichi, Osawa Satoko, Isshiki Hayato, Hori Yukiko, Shimada Naoaki, Higo Takuya, Yokoshima Satoshi, Fukuyama Tohru, Lee Virginia M. -Y., Trojanowski John Q., Tomita Taisuke, Iwatsubo Takeshi
JOURNAL OF NEUROSCIENCE Vol. 31 ( 18 ) page: 6850-6857 2011.5
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A Practical Synthesis of (-)-Kainic Acid Reviewed
Takita Satoshi, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 13 ( 8 ) page: 2068-2070 2011.4
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Concise Total Synthesis of (+)-Lyconadin A Reviewed
Nishimura Takuya, Unni Aditya K., Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 133 ( 3 ) page: 418-419 2011.1
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Let's Challenge Reviewed
Yokoshima Satoshi
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN Vol. 68 ( 12 ) page: 1323-1324 2010.12
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Development of photoaffinity probes for gamma-secretase equipped with a nitrobenzenesulfonamide-type cleavable linker (vol 19, pg 6869, 2009) Reviewed
Yokoshima Satoshi, Abe Yuzo, Watanabe Naoto, Kita Yoichi, Kan Toshiyuki, Iwatsubo Takeshi, Tomita Taisuke, Fukuyama Tohru
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 20 ( 5 ) page: 1798-1799 2010.3
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Total Synthesis of (-)-Mersicarpine Reviewed
Nakajima Rie, Ogino Tsuyoshi, Yokoshima Satoshi, Fukuyama Tohru
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 132 ( 4 ) page: 1236-+ 2010.2
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Total Synthesis of (-)-Morphine Reviewed
Koizumi Hifumi, Yokoshima Satoshi, Fukuyama Tohru
CHEMISTRY-AN ASIAN JOURNAL Vol. 5 ( 10 ) page: 2192-2198 2010
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Total Synthesis of (+)-Vinblastine: Control of the Stereochemistry at C18 ' Reviewed
Yokoshima Satoshi, Tokuyama Hidetoshi, Fukuyama Tohru
CHEMICAL RECORD Vol. 10 ( 2 ) page: 101-118 2010
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Development of photoaffinity probes for gamma-secretase equipped with a nitrobenzenesulfonamide-type cleavable linker Reviewed
Yokoshima Satoshi, Abe Yuzo, Watanabe Naoto, Kita Yoichi, Kan Toshiyuki, Iwatsubo Takeshi, Tomita Taisuke, Fukuyama Tohru
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 19 ( 24 ) page: 6869-6871 2009.12
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Total Synthesis of (-)-Huperzine A Reviewed
Koshiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 11 ( 22 ) page: 5354-5356 2009.11
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A practical synthesis of (-)-oseltamivir Reviewed
Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
TETRAHEDRON Vol. 65 ( 16 ) page: 3239-3245 2009.4
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SYNTHETIC STUDIES TOWARD (+)-LYSERGIC ACID: CONSTRUCTION OF THE TETRACYCLIC ERGOLINE SKELETON Reviewed
Inoue Tohru, Yokoshima Satoshi, Fukuyama Tohru
HETEROCYCLES Vol. 79 page: 373-378 2009.4
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TOTAL SYNTHESIS OF (+/-)-MORPHINE Reviewed
Uchida Kenji, Yokoshima Satoshi, Kan Toshiyuki, Fukuyama Tohru
HETEROCYCLES Vol. 77 ( 2 ) page: 1219-1234 2009.2
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A SIMPLE CHIRAL TEMPLATE FOR THE SYNTHESIS OF FUNCTIONALIZED alpha-ARYLGLYCINE DERIVATIVES Reviewed
Nakata Hiyoku, Imai Takahiro, Yokoshima Satoshi, Fukuyama Tohru
HETEROCYCLES Vol. 76 ( 1 ) page: 747-757 2008.9
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(1-nosyl-5-nitroindol-3-yl)methyl ester: A novel protective group for carboxylic acids Reviewed
Nishimura Takuya, Yamada Kouhei, Takebe Tohru, Yokoshima Satoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 10 ( 12 ) page: 2601-2604 2008.6
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Synthesis of eudistomin C and E: Improved preparation of the indole unit Reviewed
Yamagishi Hiroaki, Matsumoto Koji, Iwasaki Kotaro, Miyazaki Tohru, Yokoshima Satoshi, Tokuyama Hidetoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 10 ( 12 ) page: 2369-2372 2008.6
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Oseltamivir enhances hippocampal network synchronization Reviewed
Usami Atsushi, Sasaki Takuya, Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru, Yamatsugu Kenzo, Kanai Motomu, Shibasaki Masakatsu, Matsuki Norio, Ikegaya Yuji
JOURNAL OF PHARMACOLOGICAL SCIENCES Vol. 106 ( 4 ) page: 659-662 2008.4
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Oseltamivir induces spike synchronization in hippocampal networks Reviewed
Usami Atsushi, Sasaki Takuya, Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru, Yamatsugu Kenzo, Kanai Motomu, Shibasaki Masakatsu, Matsuki Norio, Ikegaya Yuji
JOURNAL OF PHARMACOLOGICAL SCIENCES Vol. 106 page: 173P-173P 2008
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Synthesis of (+)-vinblastine and its analogues Reviewed
Miyazaki Tohru, Yokoshirna Satoshi, Simizu Siro, Osada Hiroyuki, Tokuyama Hidetoshi, Fukuyama Tohru
ORGANIC LETTERS Vol. 9 ( 23 ) page: 4737-4740 2007.11
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A practical synthesis of (-)-Oseltamivir Reviewed
Satoh Nobuhiro, Akiba Takahiro, Yokoshima Satoshi, Fukuyama Tohru
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 46 ( 30 ) page: 5734-5736 2007
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Diastereoselective synthesis of atropisomeric 3-(2-substituted aryl)quinazolin-4-ones and their stereochemical properties Reviewed
Tokitoh Takashi, Kobayashi Toshitake, Nakada Eisuke, Inoue Tohru, Yokoshima Satoshi, Takahashi Hideyo, Natsugari Hideaki
HETEROCYCLES Vol. 70 page: 93-+ 2006.12
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Total synthesis of (+/-)-morphine Reviewed
Uchida Kenji, Yokoshima Satoshi, Kan Toshiyuki, Fukuyama Tohru
ORGANIC LETTERS Vol. 8 ( 23 ) page: 5311-5313 2006.11
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Synthesis of biotinylated photoaffinity probes based on arylsulfonamide gamma-secretase inhibitors Reviewed
Fuwa Haruhiko, Hiromoto Kenichi, Takahashi Yasuko, Yokoshima Satoshi, Kan Toshiyuki, Fukuyama Tohru, Iwatsubo Takeshi, Tomita Taisuke, Natsugari Hideaki
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 16 ( 16 ) page: 4184-4189 2006.8
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Novel gamma-secretase inhibitors discovered by library screening of in-house synthetic natural product intermediates Reviewed
Takahashi Y, Fuwa H, Kaneko A, Sasaki M, Yokoshima S, Koizumi H, Takebe T, Kan T, Iwatsubo T, Tomita T, Natsugari H, Fukuyama T
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 16 ( 14 ) page: 3813-3816 2006.7
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Stereocontrolled total synthesis of (+)-vincristine Reviewed
Kuboyama T, Yokoshima S, Tokuyama H, Fukuyama T
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA Vol. 101 ( 33 ) page: 11966-11970 2004.8
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A novel palladium-catalyzed coupling of thiol esters with 1-alkynes Reviewed
Tokuyama H, Miyazaki T, Yokoshima S, Fukuyama T
SYNLETT ( 10 ) page: 1512-1514 2003.8
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Stereocontrolled total synthesis of (+)-vinblastine Reviewed
Yokoshima S, Ueda T, Kobayashi S, Sato A, Kuboyama T, Tokuyama H, Fukuyama T
PURE AND APPLIED CHEMISTRY Vol. 75 ( 1 ) page: 29-38 2003.1
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Reduction of ethanethiol esters to aldehydes Reviewed
Tokuyama H, Yokoshima S, Lin SC, Li LP, Fukuyama T
SYNTHESIS-STUTTGART ( 8 ) page: 1121-1123 2002.6
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Stereocontrolled total synthesis of (+)-vinblastine Reviewed
Yokoshima S, Ueda T, Kobayashi S, Sato A, Kuboyama T, Tokuyama H, Fukuyama T
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol. 124 ( 10 ) page: 2137-2139 2002.3
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A novel oxidative transformation of alpha-aminonitriles to amides Reviewed
Yokoshima S, Kubo T, Tokuyama H, Fukuyama T
CHEMISTRY LETTERS ( 2 ) page: 122-123 2002.2
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Dogger Bank Itch revisited: isolation of (2-hydroxyethyl) dimethylsulfoxonium chloride as a cytotoxic constituent from the marine sponge Theonella aff. mirabilis Reviewed
Warabi K, Nakao Y, Matsunaga S, Fukuyama T, Kan T, Yokoshima S, Fusetani N
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY B-BIOCHEMISTRY & MOLECULAR BIOLOGY Vol. 128 ( 1 ) page: 27-30 2001.1
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Enantioselective total synthesis of (+)-gelsemine: Determination of its absolute configuration Reviewed
Yokoshima S, Tokuyama H, Fukuyama T
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION Vol. 39 ( 22 ) page: 4073-4075 2000
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A novel ketone synthesis by a palladium-catalyzed reaction of thiol esters and organozinc reagents Reviewed
Tokuyama H, Yokoshima S, Yamashita T, Fukuyama T
TETRAHEDRON LETTERS Vol. 39 ( 20 ) page: 3189-3192 1998.5
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Facile palladium-mediated conversion of ethanethiol esters to aldehydes and ketones Reviewed
Tokuyama H, Yokoshima S, Yamashita T, Lin SC, Li LP, Fukuyama T
JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY Vol. 9 ( 4 ) page: 381-387 1998