Organization
Research Institute of Environmental Medicine Designated assistant professor
Title
Designated assistant professor
KAWAMURA Kiyoshi
Degree 1
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修士（工学） （ 1994.3 名古屋工業大学 ）
Research Interests 1
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創薬化学 ドラッグディスイカバリー
Papers 9
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Systematic asymmetric analog synthesis of fluspidine, a σ1 receptor ligand, to improve ligand affinity
Tetrahedron Letters 2021.7
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Identification of a novel 2-pyridyl-benzensulfonamide derivative, RQ-00203078, as a selective and orally active TRPM8 antagonist
Bioorganic & Medicinal Chemistry Letters 2014.10
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Effects of 5-HT2B, 5-HT3 and 5-HT4 receptor antagonists on gastrointestinal motor activity in dogs
World Journal of Gastroenterology 2013.10
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Synthesis and SAR of heteroaryl-phenyl-substituted pyrazole derivatives as highly selective and potent canine COX-2 inhibitors
Bioorganic & Medicinal Chemistry Letters 2006.2
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Optimization of imidazole 5-lipoxygenase inhibitors and selection and synthesis of a development candidate
Chemical and Pharmaceutical Bulletin 2005.8
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Efficient synthesis of 4-(3-fluoro-5-{[4-(2-methyl-1H-imidazol-1-yl)benzyl]-oxy}phenyl)tetrahydro-2H-pyran-4-carboxamide, a novel 5-lipoxygenase inhibitor
Synthesis 2004.8
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Synthesis of 2-acylindole-3-acetic acids: a novel base-mediated indole synthesis
Tetrahedron Letters 2003.8
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Preparation of Optically Pure Propargylic and Allylic Alcohols from 2-(Trimethylsilyl)vinyl Sulfoxides as a Chiral Ethynyl Anion Synthon: Computational Studies on Elimination Reaction of 2-(Trimethylsilyl)vinyl Sulfoxides
Journal of Organic Chemistry 2002.1
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Convenient preparation of optically pure propargylic alcohols using 2-(trimethylsilyl)vinyl sulfoxide as a novel chiral synthon
Tetrahedron Letters 2001.5